What is Cyproterone compound for?

Cyproterone Compound is a hormonal drug that has contraceptive effects and is also used to treat skin problems such as acne. This medicine must be used under the supervision of a doctor. Cyproterone Compound tablets have other uses that we will introduce you to in this article.
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Pharmaceutical forms of cyproterone compound
This drug is sold in the form of tablets. This pill contains 2 mg of cyproterone acetate and 35 micrograms of ethinyl estradiol.
Uses of cyproterone compound
This medicine can be used in the following cases:
- Treatment of severe and resistant acne with antibiotics
- Contraception
- Help to treat ovarian laziness
- Treatment of hirsutism or hairiness in women
- Effective in the treatment of prostate cancer
Pharmacological effects and mechanism of action of Cyproterone compound
Cyproterone compound contains two components: an antiandrogen component, which is cyproterone, and an estrogenic component, which is called ethinyl estradiol. Since this medicine is in conflict with the effects of androgens, for this reason it reduces the secretion of sebum (helping to treat severe and resistant acne) and also controls the growth of extra hair. Cyproterone Acetate is an antagonist of androgen receptors and blocks androgen receptors and inhibits the release of gonadotropins from the pituitary gland. Ethinylestradiol mimics the effects of endogenous estrogen.
The dosage of Cyproterone compound
The period of taking cyproterone compound tablets is 21 days. 1 tablet should be taken daily. After 21 days of taking the pill, this pill should not be used for another 7 days. The next period starts on the eighth day and this medicine must be used again for 21 days. Of course, keep in mind that the dosage and how to use this medicine must be determined by the doctor.
Time to take cyproterone compound tablets
The time of taking Cyproterone Compound should be determined by the attending physician, but in general, it can be said that it is better to start taking it from the first day of the period. Take this tablet with 1 glass of water between meals.
What is the difference between LD and cyproterone compound?
Cyproterone compound and LD tablets differ from each other in terms of ingredients and active ingredients. LD pill is a hormonal and contraceptive drug containing levonorgestrel and ethinyl estradiol; While cyproterone and estrogen have been used in cyproterone compound. In general, both of those pills can be used to prevent pregnancy. Which one is best for you should be determined by your doctor.
Precautions
At the time of taking this pill, if symptoms of blood clot formation are observed, the use of the drug should be stopped and a doctor should be consulted. The most important of these symptoms are:
- Chest pain
- Severe and sudden cough
- Severe and prolonged headache
- Double vision or visual impairment
- Severe pain in the abdomen and leg swelling
- Inability to speak or changes in the sense of sight, smell, or taste
The use of this medicine in women smokers increases the risk of arterial diseases.
People who are overweight or have high blood pressure should use this medicine with caution.
Before using this medicine, inform your doctor if you are suffering from a certain disease and you are taking a certain medicine.
Discontinue this medication 4 to 6 weeks before surgery.
Do a Pap smear test regularly.
While taking this medicine, check your breasts every month and see a doctor if you see or feel any kind of special case (such as a lump).
Contraindications for Cyproterone Compound tablets
Cyproterone compound is contraindicated in the following cases:
- If there is a family history of these diseases under the age of 45: Varicose veins, severe depression, sickle cell anemia and inflammatory bowel diseases such as Crohn’s disease.
- If you have these problems: thrombotic disorders or history thereof, acute migraine, liver diseases, hepatitis, gallstones, history of urticaria, breast or genital carcinoma.
- In case of pregnancy
Cyproterone compound side effects
Relatively common side effects of this drug include the following:
- Varicose veins and edema
- Headache and dizziness
- Nervousness and depression
- Occurrence of pregnancy spots
- Change in libido
- Nausea and digestive problems
- Pain during menstruation
- Sensitivity to the touch of the breast
- Increased risk of genital tract infections
Does taking cyproterone compound tablets cause obesity?
Yes; This drug is one of the contraceptive drugs and in some people it may be associated with overweight and obesity. Birth control pills, especially at the beginning of use, may cause obesity and water retention in the body. If you notice an increase in weight after taking this medicine, consult your doctor.
Be careful that birth control pills do not directly cause obesity, but they may affect the appetite of some people and lead to changes in weight.
Drug interaction of cyproterone compound
Cyproterone compound interacts with the following drugs:
- Combined hepatitis C antiviral products
- Anastrazole
- Kanivaptan
- Potassium bitartrate
- Tranxamic acid
- Lactic acid and citric acid
Also, these drugs may reduce the effect of cyproterone compound:
- aprepitant, armudafinil, barbiturates, asonapravir, senobamate, enzalutamide, mitotane, rifamycin, rufinamide, phenytoin and many other drugs.
The above list is not complete. In general, before taking cyproterone compound, you should provide your doctor with a list of all your medications, even vitamins and herbal medicines, so that he can perform the necessary checks in terms of drug interactions. Also, be careful that drinking alcohol may reduce the effects of this drug.
Cyproterone compound consumption during pregnancy and breastfeeding
This drug is included in group X drugs for pregnancy. This means that its use during pregnancy is generally prohibited and may harm the fetus. During breastfeeding, you are only allowed to take this medicine on the recommendation of a doctor, which of course is not usually prescribed during this period.
Storage conditions of Cyproterone compound
- This medicine should be stored at a temperature of 15 to 30 degrees Celsius.
- There is no need to refrigerate this medicine.
Cyproterone compounds
Two compounds are used in this medicine:
- Cyproterone Acetate
- Ethinylestradiol
A final word about cyproterone compound
Cyproterone compound pill is a hormonal pill and is considered as a contraceptive pill. In this article from the online positive green pharmacy magazine, we have provided you with a complete description of this drug. In cases where acne is very severe and resistant to antibiotic treatment, this drug may be prescribed. Also, for hair growth in women, doctors may recommend this drug.
Site source: mayoclinic